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YDL223C (HBT1) gaosi pa'u CAS Numera: 489408-02-8 99% mama min.mo mea faaopoopo

Fa'amatalaga Puupuu:

HBT1 e fusifusia i le ligand-binding domain o le α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor (AMPA-R) i se faiga faʻalagolago i le glutamate.


Fa'amatalaga Oloa

Faailoga o oloa

Fua Fa'atatau

Igoa o oloa

HBT1

Isi igoa

YDL223C

CAS Nu.

489408-02-8

fua mole

C16H17F3N4O2S

mamafa mole

386.40

Mama

99.0%

Fa'aaliga

Malosi samasama malamalama

afifiina

1kg i le taga 25kg i le pa'u

Fa'aaogāga

nootropics

Folasaga o oloa

HBT1 e fusifusia i le ligand-binding domain o le α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor (AMPA-R) i se faiga faʻalagolago i le glutamate.O lona uiga o le HBT1 o se mole e mafai ona fusifusia i nofoaga patino i luga o le porotini AMPA-R pe a iai le glutamate, ma o lenei fusi e fesoasoani e faʻatonutonu le gaioiga o le porotini.O faʻamatalaga AMPA o loʻo faʻaalia i totonu o le fatugalemu o le tino ma taʻalo taua i fesoʻotaʻiga neuronal, gaioiga faʻalogo, ma aʻoaʻoga, manatua, ma synaptic plasticity.O talitali a le AMPA e tele sao i le neurotransmission faʻamalosi, faʻatalanoaina vave, faʻavavevave faʻafefeteina le tele o synapses, ma o loʻo aʻafia i tali vave a vaega synaptic i le glutamate.AMPA faʻafeiloaʻi e masani ona faʻapipiʻi faʻatasi ma NMDA faʻafeiloaʻi i synapses, ma faʻatasi latou te faʻalauteleina faiga faʻapipiʻi synaptic e aofia i le aʻoaʻoina, manatua, excitotoxicity, ma le neuroprotection.

Fa'aaliga

O le neurotrophic factor e maua mai i le faiʻai (BDNF) o se vaega neurotrophic lea e taua tele i le tausiga ma le faʻalauteleina o neu, ma e malosi ma tele aʻafiaga i luga o le faʻateleina, faʻavasegaina, ola ma le oti o sela neuronal ma non-neuronal, Galuega e pei o. se neurotransmitter modulator ma fesoasoani i le palasitika neuronal mo le aʻoaʻoina ma le manatua.O lea e taua tele mo le soifua maloloina ma le soifua manuia o le neura.Ole fa'atuputeleina ole BDNF e mafai ona fesoasoani ile togafitiga ma le puipuia o le tele o fa'ama'i.

Talosaga

O le HBT1 o se tala fou AMPA e faʻaleleia le faʻaleleia ma le maualalo o le agonism pe a faʻatusatusa i le LY451395 ma le OXP1, e faʻaosofia ai le gaosiga o le neurotrophic factor (BDNF), ma e faʻaalia ai se aafiaga itiiti i neu muamua Agitation.HBT1 fusifusia i le ligand-binding domain o le AMPA-R i se glutamate-faalagolago.Faʻatasi, latou te faʻalauiloaina faiga faʻapipiʻi synaptic e aofia i le aʻoaʻoina, manatua, faʻafiafiaga ma le neuroprotection.E mafai ona faʻaleleia atili le mafaufau ma le manatua o le faiʻai, ma faʻaleleia atili ai le aʻoaʻoina o tagata.


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