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Nefiracetam pa'u gaosi oloa CAS Numera: 77191-36-7 99% mama min.mo mea faaopoopo

Fa'amatalaga Puupuu:

O le Nefiracetam o loʻo i totonu o le vasega e faʻaleleia ai le atamai e le o tuaoi, o loʻo i ai ni vailaʻau eseese ma faʻaleleia ai le mafaufau ma puipuia le faʻaleagaina o le aʻoaʻoina ma le manatua e ala i o latou aʻafiaga i le cerebral cortex.


Fa'amatalaga Oloa

Faailoga o oloa

Fua Fa'atatau

Igoa o oloa

Nefiracetam

Isi igoa

n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamide;NEFIRACETAM;

2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide;

dm9384;

n-(2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid;DM-9384,(2-(2-Oxopyrrolidin-1-yl) -N-(2,6-dimethylphenyl) -acetamide);

DMMPA

CAS Nu.

77191-36-7

fua mole

C14H18N2O2

mamafa mole

246.3

Mama

99.0%

Fa'aaliga

Pa'epa'e pa'epa'e

afifiina

25 kilokalama/paila

Fa'aaogāga

nootropic

Folasaga o oloa

O le Nefiracetam o loʻo i totonu o le vasega e faʻaleleia ai le atamai e le o tuaoi, o loʻo i ai ni vailaʻau eseese ma faʻaleleia ai le mafaufau ma puipuia le faʻaleagaina o le aʻoaʻoina ma le manatua e ala i o latou aʻafiaga i le cerebral cortex.E leai ni mea totino a le muscarinic receptor agonists ma antagonists, e le taofia foi le gaioiga a Ach.O aʻafiaga o le faʻagaloina ma le faʻaleleia o mafaufauga o lenei vailaʻau e maua e ala i le faʻaleleia o le faʻamalolo o le Ach i le cerebral cortex.O kinase protein e faalagolago i tolauapiga e faʻaleleia ai le gaioiga o le Ca2 +, lea e ono nafa ma le faʻaleleia o le faʻamalolo o le Ach.Nefiracetam (NEF) o se pyrrolidone type nootropic agent faʻatasi ai ma vailaʻau eseese faʻapea foʻi ma le faʻaleleia o aʻafiaga.I le faoa faamalosi o le amygdala, o le nefiracetam e taofia uma ai le electroencephalographic ma amioga.O le NEF e iai se alaleo fa'ama'i fa'ama'i.

Fa'aaliga

Nefiracetam e faʻaaogaina e togafitia ai faʻamaʻi o le cerebrovascular.E mafai ona faʻaleleia le malosi o le mafaufau ma puipuia le faʻaleagaina o le aʻoaʻoina ma le manatua e ala i lona aafiaga ile cerebral cortex.E leai ni meatotino a le muscarinic receptor agonist ma le antagonistic agent, e le taofia foi le gaioiga o le acetyl cholinase.O le mea lea, o ona aʻafiaga o le faʻagaloina ma le faʻaleleia o mafaufauga e tupu e ala i le faʻaleleia o le tuʻuina atu o le acetylcholine i le cerebral cortex.

Talosaga

O le Nefiracetam o se mea e maua mai i le hydrophobic o le piracetam ma se faʻasologa faʻapipiʻi o mea uma o le Racetam piracetam.Nefiracetam o loʻo gaosia muamua e Daiichi Sankyo (kamupani vailaʻau Iapani) mo togafitiga o le AD.I le faaopoopo atu i auala uma e mafua mai i le Nefiracetam, e masani ona manatu o se mea e nafa ma le mauaina o ala o le calcium i totonu o le tino, faʻapea foʻi ma le faʻafeiloaʻi tuusaʻo o le mea e faʻaalia ai le faʻalavelave, e fai ma vaega o le agonist o le glycine-binding site o le NDMA receptor.


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