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Amino Tadalafil paʻu gaosi oloa CAS Numera: 385769-84-6 98% mama min.mo mea faaopoopo

Fa'amatalaga Puupuu:

Amino Tadalafil o se tuufaatasiga tutusa ma Tadalafil, faatasi ai ma nisi o vaega galue i lona fausaga ua suia e vaega amino.


Fa'amatalaga Oloa

Faailoga o oloa

Fua Fa'atatau

Igoa o oloa

Amino Tadalafil

Isi igoa

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3] ,4-b]indole-1,4(6H,7H)-dione

CAS Nu.

385769-84-6

fua mole

C21H18N4O4

mamafa mole

390.39

Mama

98.0%

Fa'aaliga

Pa'epa'e i le pa'epa'e pa'epa'e

Fa'aaogāga

Mea'ai Fa'aopoopo Mea'ai

Folasaga o oloa

Amino Tadalafil o se tuufaatasiga tutusa ma Tadalafil, faatasi ai ma nisi o vaega galue i lona fausaga ua suia e vaega amino.O le PDE5 inhibitor ma e iai aʻafiaga faʻafomaʻi e tutusa ma Tadalafil.E masani ona faʻaaogaina mo le togafitia o le male erectile dysfunction (ED).Pe a faʻatusatusa i Tadalafil, Amino Tadalafil e faʻagesegese le fua o le metabolic i totonu o le tino, ma e mafai ona i ai se aafiaga umi.

Fa'aaliga

(1) Filifiliga maualuga: Amino Tadalafil e maualuga le filifilia mo PDE5, faʻatasi ai ma le maualuga maualuga o le vavalalata mo PDE5 nai lo isi PDE subtypes.O lona uiga e mafai e Amino Tadalafil ona sili atu ona poloka le gaioiga o le enzyme PDE5, faʻaleleia le toto i totonu o totoga o tama tane ma faʻaleleia ai faʻamaoniga o le erectile dysfunction (ED).

(2) Aʻafiaga umi: Amino Tadalafil e faʻagesegese le metabolism i totonu o le tino, lea e mafai ai ona maua se faʻamaʻi faʻamaʻi umi, e oʻo atu i 36 itula.O le mea lea e avea ai Amino Tadalafil o se vailaʻau togafitiga ED umi, lea e le manaʻomia ona ave soo.

(3) Faʻaitiitia aʻafiaga: Amino Tadalafil e itiiti aʻafiaga e faʻatusatusa i Tadalafil, e pei o le ulu o le ulu, ma le faʻafitauli o le manava.Ona o le maualuga o le filifilia, Amino Tadalafil e mafai ona sili atu ona aloese mai fegalegaleaiga ma isi PDE subtypes, faʻaitiitia ai le aʻafiaga o aʻafiaga.

(4) Faʻamoemoega lautele: I le faaopoopo atu i le togafitia o le ED, e mafai foi ona faʻaaogaina Amino Tadalafil e togafitia ai isi faʻamaʻi e pei o le toto maualuga o le pulmonary arterial.Ole mea lea e maua ai e Amino Tadalafil avanoa faʻaoga lautele i le lumanaʻi.

Talosaga

Amino Tadalafil o se tuufaatasiga na atiae i tausaga talu ai nei, o loʻo i ai se fausaga e tutusa ma Tadalafil, ae o nisi vaega i lona fausaga ua suia e vaega amino.I le taimi nei, e leʻi faʻatagaina Amino Tadalafil mo le faʻaaogaina faafomaʻi, o lona uiga o lona faʻaaogaina i le falemaʻi e faʻatapulaʻaina.Ae ui i lea, o nisi suʻesuʻega ua faʻaalia ai o lenei tuufaatasiga e tele lona gafatia mo le faʻaaogaina.

Amino Tadalafil o le PDE5 inhibitor, lea e iai lona aafiaga faʻafomaʻi tutusa e pei o Tadalafil.E mafai ona faʻaleleia faʻamaoniga o le erectile dysfunction (ED) e ala i le faʻaleleia o le toto i totonu o totoga fanau tama e ala i le taofia o le gaioiga o le enzyme PDE5.Pe a faʻatusatusa i le Tadalafil, Amino Tadalafil e faʻagesegese le metabolism i totonu o le tino, atonu e sili atu lona aʻafiaga.O le mea lea e maua ai e Amino Tadalafil le malosi tele i le togafitiga o ED.

E le gata i lea, e mafai foi ona faʻaaogaina Amino Tadalafil e togafitia ai isi faʻamaʻi, e pei o le toto maualuga o le pulmonary arterial.O nisi suʻesuʻega ua faʻaalia ai e mafai e le iniseti PDE5 ona faʻalauteleina aʻa toto pulmonary, ma faʻaleleia ai faʻamaoniga o tagata mamaʻi e maua i le toto maualuga.Talu ai o Amino Tadalafil e iai sona aafiaga faʻafomaʻi tutusa e pei o Tadalafil, e mafai foi ona faʻaaogaina e togafitia ai le toto maualuga o le pulmonary.

I le aotelega, o Amino Tadalafil e tele lona faʻaogaina, ae sili atu suʻesuʻega faʻapitoa e manaʻomia e fuafua ai lona saogalemu ma le aoga.Afai o nei faʻataʻitaʻiga e maua ai iʻuga lelei, e mafai e Amino Tadalafil ona avea ma vailaʻau fou mo togafitiga o le ED ma le toto maualuga o le pulmonary, e maua ai le tele o togafitiga mo fomaʻi ma gasegase.


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